Benzocainum

Benzocainum Uses, Dosage, Side Effects, Mechanism of Action, How Long Does it Take to Work? Benzocainum is a brand name. Its generic name is Benzocaine.

Benzocainum

Benzocainum is a local anesthestic that is used to numb various areas of the body.

Uses For Benzocainum

Benzocainum is primarily used to relieve pain and itching from various conditions such as mouth ulcers, sore throats, teething in infants, genital itching, and hemorrhoids.

Mechanism of Action

The active ingredient in benzocaine blocks nerve signals in the body, reducing the sensation of pain and itching in the affected area. It does not reduce inflammation or swelling.

How Long Does it Take to Work?

The effects of benzocaine are almost immediate, taking about one to five minutes for the numbing sensation to kick in. The duration of the effects can last from 20-40 minutes.

Absorption

Benzocainum is absorbed through the skin, and is also known to be absorbed through ingestion.

Route of Elimination

Benzocainum is metabolized by the liver and excreted through the kidneys.

Dosage

The usual dose for adults is 5-20 milligrams applied topically, repeat as necessary. The exact dose determined by a healthcare provider depending on the condition being treated.

Administration

Benzocainum is applied topically on the affected area. It can also be ingested as a lozenge or throat spray.

Side Effects

• Allergic reactions
• Skin rash
• Hives
• Breathing difficulty
• Swelling of the face and tongue
• Loss of sensation
• Stomach upset

Toxicity

The toxic effects of benzocaine is rare and mostly seen in people who have been exposed to large doses of benzocaine. The signs of benzocaine toxicity are headache, dizziness, coma, seizures, low blood pressure, and breathing difficulties.

Precautions

• Do not use on large areas of the body
• Do not use on broken or irritated skin
• Do not use near eyes or mucous membranes
• Do not use in children younger than two years of age
• Do not use in people who have had a history of allergic reactions to local anesthetics
• Do not use if patient is taking a MAO inhibitor

Interactions

• Cimetidine
• Monoamine Oxidase Inhibitors (MAOIs)
• Estrogens
• Probenecid
• Amphetamines

Disease Interactions

• CNS Depressants
• Renal Impairment
• Respiratory Depression
• Cardiovascular Disease
• Liver Disease
• Gallbladder Disease
• Thyroid Disease

Drug Interactions

• Xiidra (ethylcellulose)
• Xenazine
• Xyrem (sodium oxybate)
• Xigduo XR (dapagliflozin and metformin hydrochloride)
• Xtampza ER (oxycodone)
• Xanax (alprazolam)
• Xeljanz XR (tofacitinib)

Food Interactions

There are no known food interactions with benzocaine.

Pregnancy Use

Benzocainum should be avoided during pregnancy unless the benefit outweighs the risk. Talk to your doctor if you are pregnant or planning a pregnancy.

Lactation Use

It is not known if benzocaine is secreted in breast milk, so it should be avoided in nursing mothers.

Acute Overdose

Overdosage of benzocaine can cause serious side effects like arrhythmias, respiratory depression, and coma. Seek immediate medical attention if an overdose is suspected.

Contraindication

Benzocainum should not be used in people who have allergies to local anesthetics. It should also not be used in people who have kidney, liver, or cardiac problems, or in any patient with a history of anemia.

Use Directions

Always read and follow the directions provided with the medication. Use benzocaine exactly as directed. Do not apply to broken or irritated skin or near the eyes or mouth.

Storage Conditions

Benzocainum should be stored at room temperature away from light and moisture.

Volume of Distribution

The volume of distribution (Vd) for benzocaine is 0.7 L/kg.

Half Life

The half-life of benzocaine is approximately 1.6 hours.

Clearance

The clearance of benzocaine is 0.97L/hr/kg.

Here you find in details version of Benzocainum

Some Frequently Asked Questions About Benzocainum

What is Benzocainum?

Benzocainum is a local anesthetic commonly used as a topical pain reliever or in cough drops. It is the active ingredient in many over-the-counter anesthetic ointments such as products for oral ulcers. It is also combined with antipyrine to form A/B otic drops to relieve ear pain and remove earwax.

What is Benzocainum used for?

Benzocainum is used topically to reduce pain and itching associated with minor skin irritations, sore throats, sunburn, teething, hemorrhoids, and other minor injuries. It may also be used to numb the skin before certain medical procedures.

Is Benzocainum harmful?

If used as directed, benzocaine is generally considered safe. However, if it is misused or overdosed, it can be harmful. Overdose and misuse can cause serious side effects, including nausea, vomiting, difficulty breathing, dizziness, and rashes.

How is Benzocainum administered?

Benzocainum is available in the form of ointments, creams, lotions, gels, patches, sprays, lozenges, or even inhalers. The method and dose of administration may vary depending on the condition for which it is being used.

How long does Benzocainum take to work?

The effects of benzocaine are usually felt within minutes after it is applied. However, it may take more time for the full effects of benzocaine to be realized.

Can Benzocainum be taken orally?

Benzocainum is approved for use in many oral products to reduce pain and itching associated with minor oral irritations. These products typically come in the form of lozenges, sprays, or creams.

Who should not use Benzocainum?

Benzocainum should not be used by people with a known allergy to it or any of its ingredients. It should also not be used on open wounds, rashes, or in the eyes, ears, or mouth. Additionally, pregnant and nursing mothers should consult their physician before using any benzocaine product.

What are the side effects of Benzocainum?

Side effects of benzocaine can include the following: nausea, dizziness, rash, itching, difficulty breathing, swelling of the mouth or throat, vomiting, and tightness in the chest. If any of these side effects occur, stop using the product and contact a physician immediately.

Are there any special precautions to take when using Benzocainum?

Yes. Benzocainum should not be used for more than seven days in a row and at higher strengths than directed. It should never be applied to open wounds, rashes, or in the eyes, ears, or mouth. Additionally, pregnant and nursing mothers should consult their physician before using any benzocaine product.

Is Benzocainum available without a prescription?

Yes. Benzocainum is a topical anesthetic available over-the-counter without a prescription. However, it is important to read labels and follow directions for use.

Can Benzocainum be used in children?

Yes. Benzocainum can be used in children age two and older, but it should be used with caution. It is important to follow the directions on the label carefully and consult a physician before use.

Does Benzocainum cause drowsiness?

No. Benzocainum is not known to cause drowsiness. However, some of the products containing benzocaine may contain other ingredients that can cause drowsiness. It is important to read the labels of the product before using it.

What should I do if I miss a dose of Benzocainum?

If you miss a dose of benzocaine, apply the missed dose as soon as you remember. Do not apply more than the recommended dose in a single day.

Is it safe to use Benzocainum while pregnant?

It is not recommended to use benzocaine while pregnant or nursing as its safety in this population has not been established. Additionally, benzocaine should not be applied to the breasts or near the genital area of a pregnant woman.

Can Benzocainum be used for treating ear infections?

No. Benzocainum is not effective in treating ear infections. It should only be used for the relief of pain associated with minor ear irritations.

Can I use Benzocainum with other medications?

Yes. Benzocainum can be used with other medications, however, some medications may interfere with the absorption and effectiveness of benzocaine. It is important to consult your physician before combining benzocaine with any other medications.

Can Benzocainum be addictive?

No. Benzocainum is not known to be addictive. However, it should be used with caution, as continuous use may cause skin irritation or an allergic reaction.

How should I store Benzocainum?

Benzocainum should be stored in a cool, dry place, away from direct sunlight and heat. It should also be kept out of reach of children and pets.

How long does Benzocainum take to expire?

Benzocainum typically has a shelf life of three years from the date of manufacture. It is important to check the expiration date on the product before using it to make sure it is still safe to use.

Does Benzocainum have any drug interactions?

Yes. Benzocainum may interact with some medications, including anticoagulants, sedatives, and antihistamines. It is important to check with your physician before using benzocaine with any other medications.

Can Benzocainum cause skin irritation?

Yes. Benzocainum can cause skin irritation, including redness, itching, dryness, and burning. If these side effects occur, stop using the product and contact a physician immediately.

Can Benzocainum be used with other topical treatments?

Yes. Benzocainum can be used with other topical treatments, including topical antibiotics, antifungals, and corticosteroids. It is important to read the label and follow directions for use carefully.

What should I do if I experience a severe allergic reaction after using Benzocainum?

If you experience a severe allergic reaction, such as a rash, vomiting, difficulty breathing, or swelling of the face or throat, after using benzocaine, stop using the product immediately and contact your physician.

Can Benzocainum cause an increase in heart rate?

Yes. Benzocainum can cause an increase in heart rate in some people. If you experience this side effect, stop using the product and contact your physician.

Can I use Benzocainum after the expiration date?

No. Benzocainum should not be used after the expiration date as it could cause skin irritation or an allergic reaction.

Can Benzocainum be used on broken skin?

No. Benzocainum should not be used on broken skin as absorption is increased and overdose is more likely. Additionally, it should never be applied to open wounds or rashes.

Does Benzocainum cause any long-term side effects?

No. Benzocainum does not cause any long-term side effects. However, repeated or prolonged use may cause skin irritation or an allergic reaction.

Does Benzocainum cause dryness or flaking of the skin?

Yes. Prolonged or repeated use of benzocaine may cause dryness or flaking of the skin. Stop using the product and consult your physician if this occurs.

Does Benzocainum have any contraindications?

Yes. Benzocainum should not be used in people with a known allergy to it or its ingredients. It should also not be used on open wounds, rashes, or in the eyes, ears, or mouth. Additionally, pregnant and nursing mothers should consult their physician before using any benzocaine product.

How long does it take for Benzocainum to wear off?

The effects of benzocaine typically last for a few hours. However, the effects may last longer in some people.

Does Benzocainum cause any adverse reactions?

Yes. Adverse reactions to benzocaine can include nausea, dizziness, rash, itching, difficulty breathing, swelling of the mouth or throat, vomiting, and tightness in the chest. If any of these side effects occur, stop using the product and contact a physician immediately.

Can Benzocainum be used on children under the age of two?

No. Benzocainum should not be used on children under the age of two without the advice of a physician.

Can Benzocainum be injected?

No. Benzocainum is a topical anesthetic and should not be injected into the skin.

Is there an OD limit on Benzocainum?

Yes. Overdose of benzocaine can lead to serious side effects including nausea, vomiting, difficulty breathing, dizziness, and rashes. Do not use more than the recommended dose.

What should I avoid while using Benzocainum?

You should avoid exposing the treated area to extreme temperatures or direct sunlight. Additionally, you should avoid swimming or showering in hot water. Finally, you should avoid drinking alcohol while using benzocaine.

Is Benzocainum safe to use on sensitive skin?

Yes. Benzocainum is generally considered safe for use on sensitive skin. However, if you experience any irritation or an allergic reaction, stop using the product and contact your physician.

Does Benzocainum have any drug interactions?

Yes. Benzocainum may interact with some medications, including anticoagulants, sedatives, and antihistamines. It is important to check with your physician before using benzocaine with any other medications.

Are there any special instructions for applying Benzocainum?

Yes. Before applying benzocaine, the area should be cleaned, dried, and free of any broken skin or open wounds. Additionally, the product should not be applied near the eyes, ears, or mouth. It is important to follow the directions on the label before use.

Can Benzocainum cause an increase in blood pressure?

Yes. Benzocainum can cause an increase in blood pressure in some people. If you experience this side effect, stop using the product and contact your physician.

What should I do if I experience a rash or burning sensation after using Benzocainum?

If you experience a rash or burning sensation after using benzocaine, stop using the product immediately and contact your physician. Prolonged or repeated use of benzocaine may cause skin irritation or an allergic reaction.

Can Benzocainum be used on a pierced area?

No. Benzocainum should not be used on a pierced area as absorption is increased and overdose is more likely. Additionally, it should never be applied to open wounds or rashes.