Cerazette
Cerazette Uses, Dosage, Side Effects, Mechanism of Action, How Long Does it Take to Work? Cerazette is a brand name. Its generic name is Desogestrel.
Cerazette Introduction
Cerazette is a progestin hormone that is used for contraception and is a derivative of the naturally occurring hormone progesterone. It is used in the manufacture of desogestrel as an active ingredient in combination with ethinylestradiol for use in oral contraceptive tablets.
Cerazette Uses
Cerazette is primarily used for contraception and is also used to treat heavy menstrual bleeding, endometriosis, and breast pain. It is also used in combination with other hormones to treat menopausal symptoms.
Cerazette Mechanism of Action
Cerazette works by suppressing ovulation and, in cases of endometriosis, focuses on reducing the concentrations of estrogen responsible for stimulating the growth of endometrial tissue.
How Long Does it Take for Cerazette to Work?
Cerazette typically works within 24-48 hours after administration and the effects can last up to three to six months.
Cerazette Absorption
Cerazette is rapidly absorbed from the gastrointestinal tract and has a bioavailability of approximately 50-80%. The peak plasma concentration of desogestrel is achieved after approximately four to five hours.
Cerazette Route of Elimination
Cerazette is excreted via the urine and feces as metabolites. Approximately 30% is excreted in the urine, while the remainder is excreted via the feces.
Cerazette Dosage
The recommended dosage of desogestrel varies based on the indication: for contraception use, the starting dose is 30 mcg once daily for 21 consecutive days followed by a 7-day rest period. For treatment of endometriosis, the recommended dose is 30 mcg twice a day for 21 consecutive days. For treatment of PMS symptoms, the recommended dose is 30 mcg once daily for 21 consecutive days.
Cerazette Administration
Cerazette can be taken with or without food. It is recommended to take it at the same time each day to maintain effectiveness.
Cerazette Side Effects
Common side effects of desogestrel include nausea, headache, breast tenderness, bloating, and breakthrough bleeding. If any of these side effects do not improve or are bothersome, it is recommended to speak to a doctor. Rare but serious side effects include an increased risk of blood clots, stroke, and heart attack.
Cerazette Toxicity
There is no established threshold for desogestrel toxicity. However, if large doses are taken, the symptoms may be similar to those of an overdose of other steroid hormones, such as dizziness, headache, nausea, vomiting, and sluggishness.
Cerazette Precautions
Cerazette should be used with caution in women with a history of cardiovascular disease, diabetes, hypertension, liver disease, or thromboembolic disorders. Women should also not take the medication if they are pregnant or breastfeeding.
Cerazette Interactions
Cerazette interacts with certain drugs, such as anticonvulsants, protease inhibitors, certain antibiotics, antifungals, and St. John's wort. It is important to tell a doctor about any other medications being taken before starting desogestrel.
Cerazette Disease Interaction
Cerazette may interact with certain diseases, such as liver disease, cardiovascular disease, diabetes, hypertension, or thromboembolic disorders. It is important to inform a doctor of any pre-existing health conditions before starting desogestrel.
Cerazette Drug Interactions
Cerazette may interact with certain drugs and affect their metabolism or activity. These drugs include anticonvulsants, protease inhibitors, certain antibiotics, antifungals, and St. John's wort.
Cerazette Food Interactions
There are no known food interactions with desogestrel.
Cerazette Use in Pregnancy
Cerazette should not be used during pregnancy as it may cause harm to a developing fetus. Women are advised to avoid becoming pregnant while taking desogestrel.
Cerazette Use in Lactation
Cerazette should not be used during lactation as it can be passed to an infant through the breastmilk and may cause adverse effects in a nursing infant.
Cerazette Acute Overdose
If an overdose of desogestrel is suspected, seek medical attention immediately. If taken orally, the symptoms may be similar to other steroid hormones, such as dizziness, headache, nausea, vomiting, and sluggishness.
Cerazette Contraindication
Cerazette is contraindicated in women with a history of thromboembolic disorders, breast cancer, or other hormone-sensitive cancer.
Cerazette Use Directions
Cerazette should be taken as directed by a doctor. Do not increase or decrease the dose without medical advice. Follow the directions on the package insert and take the medication as prescribed.
Cerazette Storage Conditions
Cerazette should be stored at room temperature and away from light and moisture. Keep the medication out of the reach of children.
Cerazette Volume of Distribution
The volume of distribution for desogestrel is approximately 3.7 L/kg.
Cerazette Half Life
The half-life of desogestrel is approximately 17-24 hours.
Cerazette Clearance
The average clearance of desogestrel is approximately 6 L/hr/kg.
Here you find in details version of Cerazette
Some Frequently Asked Questions About Cerazette
1. What is Cerazette?
Cerazette is a form of progesterone used as a contraceptive to prevent unwanted pregnancies. It is available as a combination oral contraceptive pill, usually prescribed in combination with ethinyl estradiol.
2. How does Cerazette work?
Cerazette blocks the release of the egg during ovulation, and also thickens the cervical mucus making it more difficult for sperm to get to the egg. This makes it much more difficult for a sperm to fertilize an egg.
3. Who should not use Cerazette?
Cerazette should not be taken by women who have had a history of blood clots or other associated conditions. Women who are pregnant, breastfeeding, or expecting to become pregnant should not take Cerazette. Women who have uncontrolled hypertension, diabetes, or active liver disease should also avoid Cerazette.
4. How is Cerazette taken?
Cerazette is generally taken orally in pill form. It is important to take the pill at the same time each day, and to stay on schedule. Missing any doses may decrease the efficacy of the medication in preventing pregnancy.
5. What are some common side effects of Cerazette?
Common side effects of Cerazette include nausea, vomiting, breast tenderness, headache, changes in weight, changes in libido, and spotting. Less common side effects include dizziness, hair loss, and changes in skin tone.
6. Are there any other medications or conditions that might interact negatively with Cerazette?
Yes, there are certain medications or conditions that can interact with Cerazette. These include certain antibiotics, seizure medications, HIV medications, and tuberculosis medications. Women who have a history of blood clots or other associated medical conditions should not take Cerazette.
7. What should I do if I miss a dose of Cerazette?
If you miss a dose of Cerazette, take it as soon as you remember. If you do not remember until it is time for your next dose, just take the next dose as usual. Do not take a double dose to make up for the missed dose.
8. Are there any other methods of birth control that Cerazette can be combined with?
Yes, Cerazette can be combined with other methods of birth control such as condoms, diaphragms, and other non-hormonal contraceptives. It is important to use a back-up method of contraception if you are using Cerazette.
9. Can Cerazette be used while breastfeeding?
No, desogestrel should not be used while breastfeeding as it may reduce the amount of milk produced. It is advised to wait until after breastfeeding is finished, and then start using Cerazette.
10. How long does it take for Cerazette to become effective?
Cerazette typically becomes effective as a birth control method within 24 hours of taking the first dose. However, it is important to use a back-up method of contraception for the first seven days of taking Cerazette in order to ensure maximum protection.
11. How long does it take for the effects of Cerazette to wear off?
The effects of Cerazette typically wear off within 48 hours after the last dose is taken. It is important to remember to start taking the next packet of Cerazette on schedule in order to stay protected.
12. What are the possible risks and complications associated with taking Cerazette?
The most common risks and complications associated with taking Cerazette include an increased risk of blood clots, stroke, and heart attack. It is important for women to talk to their doctor about any medical conditions and medications they are taking in order to reduce the risk of complications.
13. Does Cerazette increase the risk of breast cancer?
No, according to the World Health Organization, Cerazette does not increase the risk of breast cancer. It is important to note that the risk of Breast Cancer increases with age, and women over the age of 35 should talk to their doctor about their birth control options.
14. How long can a woman take Cerazette?
A woman can take Cerazette for as long as she needs to in order to prevent unwanted pregnancies. However, if she experiences any side effects or complications while taking Cerazette, it is important to talk to her doctor as soon as possible.
15. Does Cerazette affect fertility?
No, Cerazette does not affect fertility. After discontinuing the use of Cerazette, the natural ovulation and fertility process should resume as normal.
16. Is Cerazette safe for women over the age of 35?
Yes, Cerazette can be taken safely by women over the age of 35, as long as they do not have any medical conditions that could put them at an increased risk of complications. It is still important to talk to a healthcare provider before starting any birth control.
17. Can Cerazette be used to treat any other medical conditions?
No, Cerazette is not recommended for the treatment of any medical condition other than contraception. Other medications or treatments should be discussed with a healthcare provider.
18. Are there any over-the-counter products that contain Cerazette?
No, Cerazette is only available with a prescription from a healthcare provider. Over-the-counter products without Cerazette may be available, but it is important to discuss your options with a healthcare provider.
19. How long will it take for the body to adjust to Cerazette?
It typically takes the body up to three months to adjust to any new medication. During the first three months, it is normal to experience some side effects such as nausea, headache, and breast tenderness.
20. Does Cerazette need to be taken with food?
No, Cerazette can be taken with or without food. However, it is important to make sure that it is taken at the same time each day in order to stay protected.
21. Does Cerazette increase the risk of depression?
There is some evidence that Cerazette can increase the risk of depression in some individuals. It is important to discuss any concerns or changes in mood with a healthcare professional.
22. Can Cerazette interact with any herbal supplements?
Yes, Cerazette can interact with certain herbal supplements, so it is important to discuss all medications and supplements with a healthcare professional before taking Cerazette.
23. Is Cerazette covered by most insurance providers?
Yes, most insurance providers recognize Cerazette as an accepted form of birth control and have plans that cover it.
24. Can Cerazette cause breakthrough bleeding?
It is possible for Cerazette to cause breakthrough bleeding. If this occurs, it is important to discuss it with a healthcare provider in order to rule out any other potential causes of the bleeding.
25. What should be done if the pills are missed or vomited after taking them?
If a dose is missed or vomited after taking it, it is important to take a precautionary method of birth control such as condoms or a diaphragm until the next packet is started. If more than one dose is missed, it is important to consult a healthcare professional.
26. Does Cerazette interact with alcohol?
No, Cerazette does not interact with alcohol, but it is still important to drink responsibly and not over-consume alcohol while on birth control.
27. Is it safe to take Cerazette while traveling?
Yes, it is safe to take Cerazette while travelling as long as you do not miss any doses. If you will be travelling across different time zones, it is important to maintain the same schedule of taking the pill.
28. Can Cerazette help with acne?
Yes, in some cases Cerazette can help with mild to moderate acne by reducing the amount of sebum produced by the skin. It is important to discuss any acne concerns with a healthcare professional.
29. Is Cerazette covered by Medicaid?
Yes, most states provide coverage for Cerazette through Medicaid. It is important to contact your local Medicaid office to discuss coverage options.
30. Is it safe to take Cerazette while breastfeeding?
No, Cerazette should not be taken while breastfeeding as it may reduce the amount of milk produced. It is advised to wait until after breastfeeding is finished, and then start using Cerazette.